单位:[1]School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 100102, China[2]Institute of Clinical Medicine, China-Japan Friendship Hospital, Beijing 100029, China[3]Institute of Basic Research in Clinical Medicine, China Academy of Chinese Medical Sciences, Beijing 100700, China[4]School of Chinese Medicine, Hong Kong Baptist University, Kowloon Tong, Hong Kong, SAR 00825, China
Quinazolinones belong to a family of heterocyclic nitrogen compounds that have attracted increasing interest because of their broad spectrum of biological functions. This review describes three types of natural quinazolinones and their synthesized derivatives and summarizes their various pharmacological activities, including antifungal, anti-tumor, anti-malaria, anticonvulsant, anti-microbial, anti-inflammatory and antihyperlipidemic activities. In addition, structure-activity relationships of quinazolinone derivatives are also reviewed.
基金:
National Science Foundation of ChinaNational Natural Science Foundation of China (NSFC) [81573569, 81470177, 81001623, 81373773]; Beijing Nova ProgramBeijing Municipal Science & Technology Commission [xx2014B073]; Beijing Natural Science FoundationBeijing Natural Science Foundation [7142144]
第一作者单位:[1]School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 100102, China
通讯作者:
通讯机构:[3]Institute of Basic Research in Clinical Medicine, China Academy of Chinese Medical Sciences, Beijing 100700, China[4]School of Chinese Medicine, Hong Kong Baptist University, Kowloon Tong, Hong Kong, SAR 00825, China[*1]Institute of Basic Research in Clinical Medicine, China Academy of Chinese Medical Sciences, Beijing 100700, China.
推荐引用方式(GB/T 7714):
He Dan,Wang Menglei,Zhao Siyu,et al.Pharmaceutical prospects of naturally occurring quinazolinone and its derivatives[J].FITOTERAPIA.2017,119:136-149.doi:10.1016/j.fitote.2017.05.001.
APA:
He, Dan,Wang, Menglei,Zhao, Siyu,Shu, Yisong,Zeng, Honglian...&Liu, Yuanyan.(2017).Pharmaceutical prospects of naturally occurring quinazolinone and its derivatives.FITOTERAPIA,119,
MLA:
He, Dan,et al."Pharmaceutical prospects of naturally occurring quinazolinone and its derivatives".FITOTERAPIA 119.(2017):136-149